Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
PIK3R1 5295 OMIPALISIB CHEMBL1236962 inhibitor ClearityFoundationBiomarkers, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R1 5295 RECILISIB CHEMBL2219421 inhibitor ChemblInteractions
PIK3R1 5295 PWT-33587 CHEMBL3545006 inhibitor ChemblInteractions
PIK3R1 5295 RG-7666 CHEMBL3545324 inhibitor ChemblInteractions
PIK3R1 5295 VOXTALISIB CHEMBL3545366 inhibitor ClearityFoundationBiomarkers, MyCancerGenome, ChemblInteractions
PIK3R1 5295 ALPELISIB CHEMBL2396661 inhibitor ClearityFoundationBiomarkers, MyCancerGenome, MyCancerGenomeClinicalTrial
PIK3R1 5295 PI-103 CHEMBL573339 inhibitor MyCancerGenome
PIK3R1 5295 BUPARLISIB CHEMBL2017974 inhibitor MyCancerGenome, ChemblInteractions
PIK3R1 5295 Panulisib CHEMBL3545322 inhibitor ChemblInteractions
PIK3R1 5295 AZD-6482 CHEMBL2165191 inhibitor ChemblInteractions
PIK3R1 5295 LY-3023414 CHEMBL3544999 inhibitor ChemblInteractions
PIK3R1 5295 GSK-2636771 CHEMBL3188551 inhibitor MyCancerGenome
PIK3R1 5295 GEDATOLISIB CHEMBL592445 inhibitor ClearityFoundationBiomarkers, MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R1 5295 APITOLISIB CHEMBL1922094 inhibitor MyCancerGenome, ChemblInteractions
PIK3R1 5295 PILARALISIB (CHEMBL3218575) CHEMBL3218575 inhibitor MyCancerGenome
PIK3R1 5295 DACTOLISIB CHEMBL1879463 inhibitor ClearityFoundationBiomarkers, MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R1 5295 PF-04691502 CHEMBL1234354 inhibitor ClearityFoundationBiomarkers, MyCancerGenome, ChemblInteractions
PIK3R1 5295 Puquitinib CHEMBL3545088 inhibitor ChemblInteractions
PIK3R1 5295 SF-1126 CHEMBL2326966 inhibitor MyCancerGenome, ChemblInteractions, DrugBank
PIK3R1 5295 WORTMANNIN CHEMBL428496 DrugBank 10592235
PIK3R1 5295 VS-5584 CHEMBL1079593 inhibitor ChemblInteractions
PIK3R1 5295 COPANLISIB CHEMBL3218576 inhibitor ClearityFoundationBiomarkers, MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R1 5295 SONOLISIB CHEMBL411907 inhibitor MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R1 5295 TASELISIB CHEMBL2387080 inhibitor ChemblInteractions
PIK3R1 5295 PILARALISIB (CHEMBL3360203) CHEMBL3360203 inhibitor ChemblInteractions
PIK3R1 5295 QUERCETIN CHEMBL50 inhibitor MyCancerGenome
PIK3R1 5295 BGT-226 (CHEMBL3545096) CHEMBL3545096 inhibitor ChemblInteractions
PIK3R1 5295 PICTILISIB CHEMBL521851 inhibitor MyCancerGenome, ChemblInteractions
PIK3R1 5295 BUPARLISIB HYDROCHLORIDE CHEMBL2364604 inhibitor MyCancerGenomeClinicalTrial
PIK3R1 5295 PA-799 CHEMBL1684984 inhibitor ChemblInteractions
PIK3R1 5295 ISOPRENALINE CHEMBL1160723 agonist DrugBank 15110780, 15618457, 15381832, 15527548, 15985706
PIK3R1 5295 DS-7423 CHEMBL3545248 inhibitor ClearityFoundationBiomarkers, ChemblInteractions
PIK3R1 5295 ZSTK-474 CHEMBL586701 inhibitor ClearityFoundationBiomarkers, ChemblInteractions
PIK3R1 5295 WX-037 CHEMBL3545385 inhibitor ChemblInteractions
PIK3R1 5295 GSK-1059615 CHEMBL3544966 inhibitor ChemblInteractions

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID