Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
GRIN1 2902 AZD8108 CHEMBL3707355 antagonist ChemblInteractions
GRIN1 2902 L-GLUTAMATE CHEMBL575060 DrugBank 17662248
GRIN1 2902 (D)-SERINE CHEMBL285123 DrugBank 17139284, 17016423, 10592235
GRIN1 2902 MORPHINE CHEMBL70 NCI 12829326
GRIN1 2902 AMANTADINE HYDROCHLORIDE CHEMBL1569 antagonist ChemblInteractions
GRIN1 2902 ORPHENADRINE (CHLORIDE) CHEMBL1201023 antagonist ChemblInteractions
GRIN1 2902 MEMANTINE CHEMBL807 TdgClinicalTrial
GRIN1 2902 ORPHENADRINE CITRATE CHEMBL1200395 antagonist ChemblInteractions
GRIN1 2902 EVT-101 (CHEMBL3545349) CHEMBL3545349 antagonist ChemblInteractions
GRIN1 2902 CNS-5161 CHEMBL41306 blocker TdgClinicalTrial, ChemblInteractions, DrugBank
GRIN1 2902 RAPASTINEL CHEMBL3544917 partial agonist TdgClinicalTrial, ChemblInteractions
GRIN1 2902 RALFINAMIDE CHEMBL2107771 antagonist ChemblInteractions
GRIN1 2902 LANICEMINE CHEMBL2107647 blocker TdgClinicalTrial, ChemblInteractions
GRIN1 2902 DELUCEMINE CHEMBL2110814 antagonist ChemblInteractions
GRIN1 2902 ORPHENADRINE CHEMBL900 TdgClinicalTrial, TEND
GRIN1 2902 CERC-301 CHEMBL2068839 antagonist ChemblInteractions
GRIN1 2902 LATREPIRDINE CHEMBL589390 TdgClinicalTrial
GRIN1 2902 GW468816 CHEMBL1207366 antagonist ChemblInteractions
GRIN1 2902 Indantadol CHEMBL3707400 antagonist TdgClinicalTrial, ChemblInteractions
GRIN1 2902 CHEMBL334533 CHEMBL334533 TdgClinicalTrial
GRIN1 2902 DIMIRACETAM CHEMBL337612 TdgClinicalTrial
GRIN1 2902 NERAMEXANE CHEMBL2110954 TdgClinicalTrial
GRIN1 2902 Radiprodil CHEMBL182066 antagonist ChemblInteractions
GRIN1 2902 ESKETAMINE HYDROCHLORIDE CHEMBL2364609 ChemblInteractions
GRIN1 2902 NERAMEXANE MESYLATE CHEMBL2106798 antagonist ChemblInteractions
GRIN1 2902 GABAPENTIN CHEMBL940 DrugBank 10781913
GRIN1 2902 CHEMBL50267 CHEMBL50267 DrugBank 10592235
GRIN1 2902 CYCLOLEUCINE CHEMBL295830 DrugBank 2170997, 2556198, 2843389, 10592235
GRIN1 2902 AGMATINE CHEMBL58343 antagonist DrugBank 9918557
GRIN1 2902 NRX-1074 CHEMBL3545230 partial agonist ChemblInteractions
GRIN1 2902 NEBOGLAMINE CHEMBL1255840 positive allosteric modulator ChemblInteractions
GRIN1 2902 AV-101 CHEMBL3545351 antagonist ChemblInteractions
GRIN1 2902 ACAMPROSATE CALCIUM CHEMBL2068724 antagonist ChemblInteractions
GRIN1 2902 MEMANTINE HYDROCHLORIDE CHEMBL1699 ChemblInteractions
GRIN1 2902 KETAMINE HYDROCHLORIDE CHEMBL1714 ChemblInteractions
GRIN1 2902 TRAXOPRODIL CHEMBL17350 antagonist ChemblInteractions
GRIN1 2902 FELBAMATE CHEMBL1094 antagonist TdgClinicalTrial, ChemblInteractions
GRIN1 2902 ESKETAMINE CHEMBL395091 ChemblInteractions
GRIN1 2902 IFENPRODIL CHEMBL305187 antagonist DrugBank 3365283
GRIN1 2902 SECOBARBITAL CHEMBL447 antagonist DrugBank 7862741
GRIN1 2902 KETOBEMIDONE CHEMBL47072 antagonist DrugBank 7624018
GRIN1 2902 PRASTERONE CHEMBL90593 agonist DrugBank 9539798
GRIN1 2902 ACETYLCYSTEINE CHEMBL600 activator DrugBank 12183209
GRIN1 2902 GAVESTINEL CHEMBL44793 antagonist DrugBank 16340185
GRIN1 2902 PHENOBARBITAL CHEMBL40 antagonist DrugBank 7862741

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID
GRIN1 rs11146020 CC + CG clozapine efficacy no Genotypes CC + CG are not associated with increased response to clozapine in people with Schizophrenia as compared to genotype GG. 21332319 827789188