Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
CHEK2 11200 AZD-7762 CHEMBL2041933 inhibitor GuideToPharmacologyInteractions
CHEK2 11200 ISOGRANULATIMIDE CHEMBL413188 inhibitor GuideToPharmacologyInteractions
CHEK2 11200 PREXASERTIB CHEMBL3544911 inhibitor GuideToPharmacologyInteractions
CHEK2 11200 OLAPARIB CHEMBL521686 CGI 26510020, 2015, 322
CHEK2 11200 PF-00477736 CHEMBL3545137 inhibitor GuideToPharmacologyInteractions
CHEK2 11200 CHEMBL1236539 CHEMBL1236539 inhibitor GuideToPharmacologyInteractions
CHEK2 11200 CHEMBL179583 CHEMBL179583 inhibitor GuideToPharmacologyInteractions
CHEK2 11200 XL-844 CHEMBL3544936 TdgClinicalTrial, DrugBank

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID