Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
CACNA1I 8911 ANANDAMIDE CHEMBL15848 channel blocker GuideToPharmacologyInteractions
CACNA1I 8911 PIMOZIDE CHEMBL1423 channel blocker GuideToPharmacologyInteractions
CACNA1I 8911 GABAPENTIN CHEMBL940 modulator ChemblInteractions
CACNA1I 8911 METHSUXIMIDE CHEMBL697 blocker ChemblInteractions, TTD
CACNA1I 8911 ETHOSUXIMIDE CHEMBL696 blocker ChemblInteractions, TTD
CACNA1I 8911 IMAGABALIN CHEMBL2103836 modulator ChemblInteractions
CACNA1I 8911 ATAGABALIN CHEMBL593430 modulator ChemblInteractions
CACNA1I 8911 VERAPAMIL CHEMBL6966 inhibitor, blocker TEND, DrugBank, TTD 17139284, 17016423
CACNA1I 8911 CHEMBL1684954 CHEMBL1684954 channel blocker GuideToPharmacologyInteractions
CACNA1I 8911 FLUNARIZINE CHEMBL30008 inhibitor TdgClinicalTrial, TEND, DrugBank 17139284, 17016423, 19582593, 11784784
CACNA1I 8911 PHENSUXIMIDE CHEMBL797 blocker ChemblInteractions
CACNA1I 8911 BEPRIDIL HYDROCHLORIDE CHEMBL1200382 blocker ChemblInteractions
CACNA1I 8911 PARAMETHADIONE CHEMBL1100 suppressor, blocker TdgClinicalTrial, ChemblInteractions, TEND, DrugBank, TTD 17139284, 17016423
CACNA1I 8911 ZONISAMIDE CHEMBL750 inhibitor TdgClinicalTrial, DrugBank 19557119, 14965331, 20025128, 18433351, 20001433, 14704463, 20502722, 15511691, 17762320, 19948168
CACNA1I 8911 PREGABALIN CHEMBL1059 modulator ChemblInteractions, TTD
CACNA1I 8911 GABAPENTIN ENACARBIL CHEMBL1628502 modulator ChemblInteractions, TTD
CACNA1I 8911 MIBEFRADIL DIHYDROCHLORIDE CHEMBL1534525 blocker ChemblInteractions
CACNA1I 8911 CINNARIZINE CHEMBL43064 inhibitor DrugBank 1281221, 3530295
CACNA1I 8911 MIBEFRADIL CHEMBL45816 inhibitor, blocker, channel blocker GuideToPharmacologyInteractions, DrugBank, TTD 9375939, 15562257, 16899990, 9481612
CACNA1I 8911 TRIMETHADIONE CHEMBL695 blocker ChemblInteractions, TTD
CACNA1I 8911 CELECOXIB CHEMBL118 PharmGKB

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID
CACNA1I rs3747178 T ethosuximide efficacy yes as measured by minor allele (T) frequency in not–seizure‐free vs seizure-free children. Allele T is associated with decreased clinical benefit to ethosuximide in children with Epilepsy as compared to allele C. 28165634 1451134046