Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
PIK3R3 8503 GSK-1059615 CHEMBL3544966 inhibitor ChemblInteractions
PIK3R3 8503 PILARALISIB (CHEMBL3360203) CHEMBL3360203 inhibitor ChemblInteractions
PIK3R3 8503 VOXTALISIB CHEMBL3545366 inhibitor MyCancerGenome, ChemblInteractions
PIK3R3 8503 BUPARLISIB HYDROCHLORIDE CHEMBL2364604 inhibitor MyCancerGenomeClinicalTrial
PIK3R3 8503 BGT-226 (CHEMBL3545096) CHEMBL3545096 inhibitor ChemblInteractions
PIK3R3 8503 ZSTK-474 CHEMBL586701 inhibitor ChemblInteractions
PIK3R3 8503 Panulisib CHEMBL3545322 inhibitor ChemblInteractions
PIK3R3 8503 SONOLISIB CHEMBL411907 inhibitor MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R3 8503 LY-3023414 CHEMBL3544999 inhibitor ChemblInteractions
PIK3R3 8503 GSK-2636771 CHEMBL3188551 inhibitor MyCancerGenome
PIK3R3 8503 PI-103 CHEMBL573339 inhibitor MyCancerGenome
PIK3R3 8503 APITOLISIB CHEMBL1922094 inhibitor MyCancerGenome, ChemblInteractions
PIK3R3 8503 GEDATOLISIB CHEMBL592445 inhibitor MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R3 8503 PWT-33587 CHEMBL3545006 inhibitor ChemblInteractions
PIK3R3 8503 ISOPRENALINE CHEMBL1160723 agonist DrugBank 15110780, 15618457, 15381832, 15527548, 15985706
PIK3R3 8503 RECILISIB CHEMBL2219421 inhibitor ChemblInteractions
PIK3R3 8503 VS-5584 CHEMBL1079593 inhibitor ChemblInteractions
PIK3R3 8503 Puquitinib CHEMBL3545088 inhibitor ChemblInteractions
PIK3R3 8503 COPANLISIB CHEMBL3218576 inhibitor MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R3 8503 BUPARLISIB CHEMBL2017974 inhibitor MyCancerGenome, ChemblInteractions
PIK3R3 8503 PF-04691502 CHEMBL1234354 inhibitor MyCancerGenome, ChemblInteractions
PIK3R3 8503 TASELISIB CHEMBL2387080 inhibitor ChemblInteractions
PIK3R3 8503 ALPELISIB CHEMBL2396661 inhibitor MyCancerGenome, MyCancerGenomeClinicalTrial
PIK3R3 8503 PILARALISIB (CHEMBL3218575) CHEMBL3218575 inhibitor MyCancerGenome
PIK3R3 8503 WX-037 CHEMBL3545385 inhibitor ChemblInteractions
PIK3R3 8503 SF-1126 CHEMBL2326966 inhibitor MyCancerGenome, ChemblInteractions, DrugBank
PIK3R3 8503 QUERCETIN CHEMBL50 inhibitor MyCancerGenome
PIK3R3 8503 DS-7423 CHEMBL3545248 inhibitor ChemblInteractions
PIK3R3 8503 RG-7666 CHEMBL3545324 inhibitor ChemblInteractions
PIK3R3 8503 PICTILISIB CHEMBL521851 inhibitor MyCancerGenome, ChemblInteractions
PIK3R3 8503 DACTOLISIB CHEMBL1879463 inhibitor MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R3 8503 OMIPALISIB CHEMBL1236962 inhibitor ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R3 8503 PA-799 CHEMBL1684984 inhibitor ChemblInteractions
PIK3R3 8503 AZD-6482 CHEMBL2165191 inhibitor ChemblInteractions

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID