Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
CXCR4 7852 FRAMYCETIN CHEMBL2104426 antagonist DrugBank 14638394, 11747436
CXCR4 7852 PHENPROCOUMON CHEMBL16694 antagonist GuideToPharmacologyInteractions
CXCR4 7852 MSX-122 CHEMBL3545330 antagonist TdgClinicalTrial, ChemblInteractions, TTD
CXCR4 7852 POL6326 CHEMBL3545105 antagonist ChemblInteractions
CXCR4 7852 CHEMBL518924 CHEMBL518924 TdgClinicalTrial, DrugBank
CXCR4 7852 ULOCUPLUMAB CHEMBL3039543 antibody TdgClinicalTrial, GuideToPharmacologyInteractions
CXCR4 7852 CTCE-9908 CHEMBL3544949 antagonist ChemblInteractions
CXCR4 7852 CHEMBL452864 CHEMBL452864 antagonist GuideToPharmacologyInteractions
CXCR4 7852 CHEMBL460491 CHEMBL460491 antagonist GuideToPharmacologyInteractions
CXCR4 7852 Burixafor CHEMBL3545224 antagonist TdgClinicalTrial, ChemblInteractions
CXCR4 7852 CHEMBL1088913 CHEMBL1088913 antagonist TTD
CXCR4 7852 BKT140 CHEMBL3545348 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions
CXCR4 7852 ROLOFYLLINE (CHEMBL52333) CHEMBL52333 agonist GuideToPharmacologyInteractions
CXCR4 7852 METHIONINE SULFOXIDE CHEMBL445753 agonist GuideToPharmacologyInteractions
CXCR4 7852 PLERIXAFOR CHEMBL18442 partial agonist, antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, DrugBank, TTD 23204107, 18847313

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID