Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
AURKA 6790 AMG-900 CHEMBL2140408 inhibitor TALC, MyCancerGenome, ClearityFoundationClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions
AURKA 6790 ORANTINIB CHEMBL274654 inhibitor TTD
AURKA 6790 TAK-901 CHEMBL3544932 inhibitor TALC, MyCancerGenome
AURKA 6790 PHENYLTHIOUREA CHEMBL263376 CIViC 27209210
AURKA 6790 BARASERTIB CHEMBL415049 inhibitor GuideToPharmacologyInteractions
AURKA 6790 CHEMBL1765740 CHEMBL1765740 inhibitor GuideToPharmacologyInteractions
AURKA 6790 PF-562271 CHEMBL1084546 inhibitor GuideToPharmacologyInteractions
AURKA 6790 MK-6592 CHEMBL3545378 inhibitor ChemblInteractions
AURKA 6790 AT-9283 CHEMBL495727 inhibitor GuideToPharmacologyInteractions, ChemblInteractions, DrugBank, MyCancerGenome, TdgClinicalTrial, TTD, TALC
AURKA 6790 CYC-116 CHEMBL482967 inhibitor TALC, TdgClinicalTrial, ChemblInteractions, DrugBank, TTD
AURKA 6790 CHEMBL495758 CHEMBL495758 DrugBank 10592235
AURKA 6790 MK-5108 CHEMBL3182444 inhibitor TALC, MyCancerGenome, GuideToPharmacologyInteractions, ChemblInteractions, TTD
AURKA 6790 CENISERTIB CHEMBL1614709 inhibitor TdgClinicalTrial, ChemblInteractions, TTD
AURKA 6790 MLN-8054 CHEMBL259084 inhibitor GuideToPharmacologyInteractions, ChemblInteractions, TTD
AURKA 6790 ANILINOQUINAZOLINE1 CHEMBL382590 inhibitor GuideToPharmacologyInteractions
AURKA 6790 CHEMBL359482 CHEMBL359482 inhibitor GuideToPharmacologyInteractions
AURKA 6790 TAS-119 CHEMBL3545326 inhibitor ChemblInteractions
AURKA 6790 RG-1530 CHEMBL1980391 inhibitor ChemblInteractions
AURKA 6790 CHEMBL223147 CHEMBL223147 DrugBank 10592235
AURKA 6790 ANILINOPYRIMIDINE1 CHEMBL383899 inhibitor GuideToPharmacologyInteractions, DrugBank 10592235
AURKA 6790 CHEMBL522891 CHEMBL522891 DrugBank 10592235
AURKA 6790 ENMD-2076 CHEMBL482968 inhibitor MyCancerGenome, GuideToPharmacologyInteractions, TdgClinicalTrial, TALC, TTD, ClearityFoundationClinicalTrial, ChemblInteractions
AURKA 6790 GSK-1070916 CHEMBL1090479 inhibitor GuideToPharmacologyInteractions
AURKA 6790 CHEMBL202721 CHEMBL202721 inhibitor GuideToPharmacologyInteractions
AURKA 6790 CHEMBL369507 CHEMBL369507 DrugBank 17139284, 17016423
AURKA 6790 ALISERTIB CHEMBL483158 inhibitor DrugBank, GuideToPharmacologyInteractions, ChemblInteractions, TALC, TTD, CancerCommons, MyCancerGenomeClinicalTrial, TdgClinicalTrial, MyCancerGenome
AURKA 6790 CHEMBL472193 CHEMBL472193 DrugBank 10592235
AURKA 6790 SNS-314 CHEMBL482767 inhibitor TALC, MyCancerGenome, TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, DrugBank, TTD 10592235
AURKA 6790 CHEMBL521105 CHEMBL521105 DrugBank 10592235
AURKA 6790 DANUSERTIB CHEMBL402548 inhibitor TALC, MyCancerGenome, GuideToPharmacologyInteractions, ChemblInteractions, TTD
AURKA 6790 PF-03814735 CHEMBL3545078 inhibitor TALC, MyCancerGenome, ChemblInteractions, TTD
AURKA 6790 TOZASERTIB CHEMBL572878 inhibitor TALC, TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TTD
AURKA 6790 XL-228 CHEMBL3545085 TdgClinicalTrial
AURKA 6790 ALISERTIB SODIUM CHEMBL2103871 ClearityFoundationClinicalTrial
AURKA 6790 TAMOXIFEN CHEMBL83 CIViC 24166501
AURKA 6790 KW-2449 CHEMBL1908397 inhibitor GuideToPharmacologyInteractions, ChemblInteractions
AURKA 6790 ENMD-981693 CHEMBL52885 inhibitor ChemblInteractions
AURKA 6790 ILORASERTIB CHEMBL1980297 inhibitor ChemblInteractions
AURKA 6790 TTP-607 CHEMBL3545327 inhibitor ChemblInteractions
AURKA 6790 FLUOROURACIL CHEMBL185 CIViC 25924824
AURKA 6790 PACLITAXEL CHEMBL428647 CIViC 12559175

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID