Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
BRCA1 672 CARBOPLATIN CHEMBL1351 ClearityFoundationBiomarkers, CKB, CIViC 25824335, 27998224, 21135055, 25847936
BRCA1 672 IROFULVEN CHEMBL118218 NCI 17229870
BRCA1 672 VINORELBINE BASE CHEMBL553025 CKB, NCI 14559807, 26801247
BRCA1 672 VELIPARIB CHEMBL506871 ClearityFoundationBiomarkers, CKB, CGI 25824335, 26842236, 26801247, 25589624
BRCA1 672 PHENYLTHIOUREA CHEMBL263376 CIViC 24240112, 21920589
BRCA1 672 TEMOZOLOMIDE CHEMBL810 CKB
BRCA1 672 TAMOXIFEN CHEMBL83 PharmGKB, NCI 15750629
BRCA1 672 GEMCITABINE CHEMBL888 NCI 12684687
BRCA1 672 MITOXANTRONE CHEMBL58 NCI 12684687
BRCA1 672 NIRAPARIB CHEMBL1094636 ClearityFoundationBiomarkers, OncoKB, CKB 27717299, 23810788, 27908594, 28229583
BRCA1 672 OLAPARIB CHEMBL521686 ClearityFoundationBiomarkers, OncoKB, CKB, CGI, CIViC 20609467, 25366685, 19553641, 20406929, 21862407, 20609468, 23346317, 28578601, 25218906, 28792849, 25193512, 27454287, 22172724, 26546619
BRCA1 672 OXALIPLATIN CHEMBL414804 ClearityFoundationBiomarkers
BRCA1 672 CHLORAMBUCIL CHEMBL515 CKB 25193512
BRCA1 672 VX-970 CHEMBL3545202 CKB
BRCA1 672 AZD-1775 CHEMBL1976040 CKB 27998224
BRCA1 672 PACLITAXEL CHEMBL428647 CKB, NCI 12684687
BRCA1 672 RUCAPARIB CHEMBL1173055 ClearityFoundationBiomarkers, OncoKB, CKB, CGI, CIViC 27908594, 27717299, 28229583, 28588062, 26779812, 27002934, 27454289
BRCA1 672 CYCLOPHOSPHAMIDE CHEMBL88 CKB 25589624
BRCA1 672 BLEOMYCIN (CHEMBL3039590) CHEMBL3039590 NCI 14559807
BRCA1 672 DOXORUBICIN CHEMBL53463 NCI 12698198
BRCA1 672 MITOMYCIN CHEMBL105 NCI 15782115
BRCA1 672 TALAZOPARIB CHEMBL3137320 ClearityFoundationBiomarkers, CKB, CIViC 28242752, 23881923, 26546619
BRCA1 672 IRINOTECAN CHEMBL481 CKB 26842236
BRCA1 672 METFORMIN CHEMBL1431 CKB 26546619
BRCA1 672 QUARFLOXIN CHEMBL2103818 CIViC 28211448
BRCA1 672 CEDIRANIB CHEMBL491473 CIViC 25218906
BRCA1 672 DENOSUMAB CHEMBL1237023 CKB 27322743
BRCA1 672 EMODIN CHEMBL289277 NCI 14694444
BRCA1 672 EVEROLIMUS CHEMBL1908360 CKB 26546619

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID