Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
AVPR1A 552 FELYPRESSIN CHEMBL1908309 agonist TdgClinicalTrial, TEND, DrugBank, TTD 18655903, 11752352, 17139284, 17016423
AVPR1A 552 TERLIPRESSIN CHEMBL2135460 stimulator TdgClinicalTrial, TEND, DrugBank, TTD 16011575, 11752352, 17303660, 16532916, 16511036, 17275806
AVPR1A 552 CHEMBL265859 CHEMBL265859 agonist GuideToPharmacologyInteractions
AVPR1A 552 CHEMBL332447 CHEMBL332447 agonist GuideToPharmacologyInteractions
AVPR1A 552 CHEMBL70099 CHEMBL70099 antagonist GuideToPharmacologyInteractions
AVPR1A 552 APRACLONIDINE CHEMBL647 antagonist GuideToPharmacologyInteractions
AVPR1A 552 MOZAVAPTAN CHEMBL420762 antagonist GuideToPharmacologyInteractions
AVPR1A 552 NELIVAPTAN CHEMBL582857 antagonist GuideToPharmacologyInteractions
AVPR1A 552 CHEMBL3307200 CHEMBL3307200 antagonist GuideToPharmacologyInteractions
AVPR1A 552 CHEMBL307483 CHEMBL307483 antagonist GuideToPharmacologyInteractions
AVPR1A 552 SELEPRESSIN CHEMBL1817709 agonist ChemblInteractions
AVPR1A 552 RG7314 CHEMBL3545342 antagonist ChemblInteractions
AVPR1A 552 VASOPRESSIN TANNATE CHEMBL1201528 agonist ChemblInteractions
AVPR1A 552 VASOPRESSIN CHEMBL373742 agonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, DrugBank 17275806, 16011575, 17303660, 16532916, 16511036
AVPR1A 552 CHEMBL435323 CHEMBL435323 agonist GuideToPharmacologyInteractions
AVPR1A 552 OXYTOCIN CHEMBL395429 agonist GuideToPharmacologyInteractions
AVPR1A 552 ATOSIBAN CHEMBL382301 antagonist GuideToPharmacologyInteractions
AVPR1A 552 APRINDINE CHEMBL1213033 antagonist GuideToPharmacologyInteractions
AVPR1A 552 CONIVAPTAN HYDROCHLORIDE CHEMBL1201108 antagonist ChemblInteractions
AVPR1A 552 DESMOPRESSIN ACETATE CHEMBL1200556 agonist ChemblInteractions, DrugBank 10731046, 8957254, 15613460, 10594321
AVPR1A 552 LYPRESSIN CHEMBL1200690 agonist ChemblInteractions
AVPR1A 552 CONIVAPTAN CHEMBL1755 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, TEND, DrugBank, TTD 16522696, 19695403, 17592003, 11752352, 17202666, 17919259, 19663609, 20054444, 17428103, 19057376
AVPR1A 552 ARGIPRESTOCIN CHEMBL2370156 agonist GuideToPharmacologyInteractions
AVPR1A 552 CHEMBL3274309 CHEMBL3274309 agonist GuideToPharmacologyInteractions
AVPR1A 552 CHEMBL296908 CHEMBL296908 antagonist GuideToPharmacologyInteractions
AVPR1A 552 MERCAPTOPURINE CHEMBL1425 antagonist GuideToPharmacologyInteractions
AVPR1A 552 SATAVAPTAN CHEMBL2107777 antagonist GuideToPharmacologyInteractions
AVPR1A 552 ANTIPYRINE CHEMBL277474 antagonist GuideToPharmacologyInteractions
AVPR1A 552 SRX251 CHEMBL3545146 antagonist ChemblInteractions
AVPR1A 552 AMSACRINE CHEMBL43 agonist GuideToPharmacologyInteractions
AVPR1A 552 CHEMBL1254024 CHEMBL1254024 antagonist GuideToPharmacologyInteractions
AVPR1A 552 RELCOVAPTAN CHEMBL419667 antagonist GuideToPharmacologyInteractions, ChemblInteractions
AVPR1A 552 ANTHRACENE-9-CARBOXYLIC ACID CHEMBL1513985 antagonist GuideToPharmacologyInteractions
AVPR1A 552 K-252A CHEMBL281948 antagonist GuideToPharmacologyInteractions
AVPR1A 552 SRX246 CHEMBL244243 antagonist ChemblInteractions
AVPR1A 552 TOLVAPTAN CHEMBL344159 antagonist GuideToPharmacologyInteractions, DrugBank 20637957

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID