Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
ATP1A1 476 DIGOXIN CHEMBL1751 inhibitor TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, DrugBank 11272406, 11309248, 11515751, 11687608, 11324464
ATP1A1 476 DIAZOXIDE CHEMBL181 other DrugBank 17287451, 12086984, 17281115
ATP1A1 476 BRETYLIUM CHEMBL1199080 inhibitor DrugBank 15121098, 1662173, 1334399, 1667290
ATP1A1 476 OUABAIN CHEMBL222863 inhibitor, binder TdgClinicalTrial, TEND, DrugBank, TTD 10564763, 10593655, 10567200, 11752352, 10541475, 10593659
ATP1A1 476 BEPRIDIL CHEMBL1008 inhibitor TdgClinicalTrial, TEND, DrugBank 2938592, 2933041, 2207500, 2148481, 1329768
ATP1A1 476 DIGITOXIN CHEMBL254219 inhibitor TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, DrugBank 11309248, 19751721, 136410, 132355, 131389, 123547
ATP1A1 476 ALMITRINE CHEMBL1183717 binder TdgClinicalTrial, TEND, DrugBank, TTD 8099718, 11752352, 2165421, 2527061, 2144185
ATP1A1 476 CHEMBL444449 CHEMBL444449 binder TTD
ATP1A1 476 POTASSIUM ACETATE CHEMBL1201058 DrugBank 17334838, 17444965, 17366541, 17347782, 17369284
ATP1A1 476 CICLOPIROX CHEMBL1413 binder TTD
ATP1A1 476 CHEMBL38827 CHEMBL38827 binder TTD
ATP1A1 476 ISTAROXIME CHEMBL3138451 TdgClinicalTrial
ATP1A1 476 HYDROFLUMETHIAZIDE CHEMBL1763 DrugBank 17139284, 17016423
ATP1A1 476 DESLANOSIDE CHEMBL1614 inhibitor, binder TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, DrugBank, TTD 11752352, 16319518
ATP1A1 476 MAGNESIUM CHEMBL2146125 DrugBank 17294093, 16928192, 16808357, 16990961
ATP1A1 476 ACETYLDIGITOXIN CHEMBL3545057 inhibitor TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, DrugBank 2826993
ATP1A1 476 TRICHLORMETHIAZIDE CHEMBL1054 inhibitor DrugBank 7752578

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID