Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
GRM5 2915 Raseglurant CHEMBL3545036 modulator TdgClinicalTrial, ChemblInteractions, DrugBank, TTD
GRM5 2915 AZD2516 CHEMBL3545346 antagonist ChemblInteractions, TTD
GRM5 2915 MAVOGLURANT CHEMBL3087515 antagonist ChemblInteractions
GRM5 2915 RUFINAMIDE CHEMBL1201754 inhibitor DrugBank 21351809
GRM5 2915 FENOBAM CHEMBL239800 modulator TTD
GRM5 2915 AZD2066 CHEMBL3545164 antagonist, modulator TdgClinicalTrial, ChemblInteractions, TTD
GRM5 2915 DIPRAGLURANT CHEMBL2346738 modulator ChemblInteractions, DrugBank, TTD
GRM5 2915 LY545694 CHEMBL3545161 antagonist ChemblInteractions
GRM5 2915 STX107 CHEMBL3545037 TdgClinicalTrial, ChemblInteractions
GRM5 2915 ACAMPROSATE CHEMBL1201293 TdgClinicalTrial
GRM5 2915 GANCICLOVIR CHEMBL182 NCI 12068048, 12231639
GRM5 2915 ALCOHOL CHEMBL545 NCI 15717208
GRM5 2915 RG7342 CHEMBL3545203 modulator ChemblInteractions
GRM5 2915 BASIMGLURANT CHEMBL3301626 modulator ChemblInteractions

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID