Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
GRIN2C 2905 D-ASPARTATE CHEMBL29757 agonist GuideToPharmacologyInteractions
GRIN2C 2905 N-METHYL-D-ASPARTIC ACID (NMDA) CHEMBL291278 agonist GuideToPharmacologyInteractions
GRIN2C 2905 MESORIDAZINE CHEMBL1088 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 LEVORPHANOL CHEMBL592 channel blocker GuideToPharmacologyInteractions
GRIN2C 2905 CNS-5161 CHEMBL41306 blocker TdgClinicalTrial, ChemblInteractions
GRIN2C 2905 RALFINAMIDE CHEMBL2107771 antagonist ChemblInteractions
GRIN2C 2905 ESKETAMINE CHEMBL395091 ChemblInteractions
GRIN2C 2905 LANICEMINE CHEMBL2107647 blocker TdgClinicalTrial, ChemblInteractions
GRIN2C 2905 ORPHENADRINE (CHLORIDE) CHEMBL1201023 antagonist ChemblInteractions
GRIN2C 2905 GLYCINE CHEMBL773 agonist GuideToPharmacologyInteractions, DrugBank 17139284, 17016423, 11861317, 8955518, 9073168
GRIN2C 2905 CHEMBL287327 CHEMBL287327 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 TENOCYCLIDINE CHEMBL279676 antagonist DrugBank 2538766
GRIN2C 2905 ESKETAMINE HYDROCHLORIDE CHEMBL2364609 ChemblInteractions
GRIN2C 2905 NEBOGLAMINE CHEMBL1255840 positive allosteric modulator ChemblInteractions
GRIN2C 2905 ACAMPROSATE CALCIUM CHEMBL2068724 antagonist ChemblInteractions
GRIN2C 2905 DELUCEMINE CHEMBL2110814 antagonist ChemblInteractions
GRIN2C 2905 (D)-SERINE CHEMBL285123 agonist GuideToPharmacologyInteractions
GRIN2C 2905 CHEMBL280828 CHEMBL280828 agonist GuideToPharmacologyInteractions
GRIN2C 2905 CHEMBL50267 CHEMBL50267 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 CONANTOKIN G CHEMBL525025 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 SELFOTEL CHEMBL39664 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 CHEMBL22304 CHEMBL22304 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 MODAFINIL CHEMBL1373 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 AMANTADINE HYDROCHLORIDE CHEMBL1569 antagonist, channel blocker GuideToPharmacologyInteractions, ChemblInteractions
GRIN2C 2905 DEXTROMETHORPHAN CHEMBL52440 channel blocker GuideToPharmacologyInteractions
GRIN2C 2905 DEXTRORPHAN CHEMBL1254766 channel blocker GuideToPharmacologyInteractions
GRIN2C 2905 DIZOCILPINE CHEMBL284237 channel blocker GuideToPharmacologyInteractions
GRIN2C 2905 MAGNESIUM CHEMBL2146125 channel blocker GuideToPharmacologyInteractions
GRIN2C 2905 CHEMBL1184349 CHEMBL1184349 channel blocker GuideToPharmacologyInteractions
GRIN2C 2905 PHENCYCLIDINE CHEMBL275528 channel blocker GuideToPharmacologyInteractions
GRIN2C 2905 PHORBOL MYRISTATE ACETATE CHEMBL279115 NCI 16417568
GRIN2C 2905 NRX-1074 CHEMBL3545230 partial agonist ChemblInteractions
GRIN2C 2905 AV-101 CHEMBL3545351 antagonist ChemblInteractions
GRIN2C 2905 Indantadol CHEMBL3707400 antagonist TdgClinicalTrial, ChemblInteractions
GRIN2C 2905 DIMIRACETAM CHEMBL337612 TdgClinicalTrial
GRIN2C 2905 KETAMINE HYDROCHLORIDE CHEMBL1714 ChemblInteractions
GRIN2C 2905 MEMANTINE HYDROCHLORIDE CHEMBL1699 ChemblInteractions
GRIN2C 2905 NERAMEXANE MESYLATE CHEMBL2106798 antagonist ChemblInteractions
GRIN2C 2905 L-GLUTAMATE CHEMBL575060 DrugBank 9417820, 17139284, 17016423, 10455281, 7905294
GRIN2C 2905 ASPARTIC ACID CHEMBL274323 agonist GuideToPharmacologyInteractions
GRIN2C 2905 CHEMBL140784 CHEMBL140784 agonist GuideToPharmacologyInteractions
GRIN2C 2905 CGP-37849 CHEMBL29811 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 CHEMBL31741 CHEMBL31741 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 CHEMBL173031 CHEMBL173031 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 CHEMBL191838 CHEMBL191838 antagonist GuideToPharmacologyInteractions
GRIN2C 2905 KETAMINE CHEMBL742 channel blocker GuideToPharmacologyInteractions
GRIN2C 2905 AZD8108 CHEMBL3707355 antagonist ChemblInteractions
GRIN2C 2905 RAPASTINEL CHEMBL3544917 partial agonist ChemblInteractions
GRIN2C 2905 FELBAMATE CHEMBL1094 antagonist ChemblInteractions
GRIN2C 2905 ORPHENADRINE CITRATE CHEMBL1200395 antagonist ChemblInteractions
GRIN2C 2905 LATREPIRDINE CHEMBL589390 TdgClinicalTrial
GRIN2C 2905 GW468816 CHEMBL1207366 antagonist ChemblInteractions

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID