Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
GABBR1 2550 PROGABIDE CHEMBL287631 agonist TdgClinicalTrial, TEND, DrugBank 2985405, 11752352, 9443561
GABBR1 2550 ARBACLOFEN PLACARBIL CHEMBL2107312 agonist ChemblInteractions, DrugBank 10494996, 11752352, 8388192, 10545129, 19303900, 10094428, 10444662, 10482760, 10386831
GABBR1 2550 SODIUM OXYBATE CHEMBL1200682 agonist ChemblInteractions
GABBR1 2550 ARBACLOFEN CHEMBL301742 agonist TdgClinicalTrial, ChemblInteractions, DrugBank 10494996, 11752352, 8388192, 10545129, 19303900, 10094428, 10444662, 10482760, 10386831
GABBR1 2550 BACLOFEN CHEMBL701 agonist TdgClinicalTrial, ChemblInteractions, NCI, TEND, DrugBank 7674378, 9486305, 10494996, 11752352, 8388192, 10545129, 19303900, 10094428, 10444662, 10482760, 10386831
GABBR1 2550 VIGABATRIN CHEMBL89598 agonist TdgClinicalTrial, DrugBank 20655489
GABBR1 2550 Lesogaberan CHEMBL448343 agonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions
GABBR1 2550 OXYBATE CHEMBL1342 TdgClinicalTrial
GABBR1 2550 CHEMBL113553 CHEMBL113553 agonist GuideToPharmacologyInteractions
GABBR1 2550 CHEMBL112797 CHEMBL112797 DrugBank

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID