Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
PARP1 142 CHEMBL401843 CHEMBL401843 DrugBank 17139284, 17016423, 10592235
PARP1 142 CHEMBL123978 CHEMBL123978 DrugBank 17139284, 17016423, 10592235
PARP1 142 CHEMBL338790 CHEMBL338790 DrugBank 10592235
PARP1 142 RUCAPARIB CHEMBL1173055 antagonist, inhibitor TALC, MyCancerGenome, ClearityFoundationClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, DrugBank
PARP1 142 CHEMBL125200 CHEMBL125200 DrugBank 17139284, 17016423, 10592235
PARP1 142 TALAZOPARIB CHEMBL3137320 inhibitor TALC, ClearityFoundationClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions
PARP1 142 RUCAPARIB CAMSYLATE CHEMBL3833368 inhibitor ChemblInteractions
PARP1 142 NIACINAMIDE CHEMBL1140 binder DrugBank, TTD 11752352
PARP1 142 CHEMBL134022 CHEMBL134022 DrugBank 10592235
PARP1 142 CHEMBL452800 CHEMBL452800 DrugBank 10592235
PARP1 142 CHEMBL361054 CHEMBL361054 DrugBank 10592235
PARP1 142 HEPTANOATE CHEMBL320358 inhibitor GuideToPharmacologyInteractions
PARP1 142 INOSINE CHEMBL1556 inhibitor TTD
PARP1 142 CHEMBL123904 CHEMBL123904 DrugBank 10592235
PARP1 142 VELIPARIB CHEMBL506871 inhibitor TALC, MyCancerGenome, ClearityFoundationClinicalTrial, ChemblInteractions, DrugBank, CancerCommons, MyCancerGenomeClinicalTrial 10592235
PARP1 142 NIRAPARIB CHEMBL1094636 inhibitor MyCancerGenome, GuideToPharmacologyInteractions, TALC, ClearityFoundationClinicalTrial, TdgClinicalTrial, TTD, ChemblInteractions
PARP1 142 INIPARIB CHEMBL1170047 inhibitor TALC, MyCancerGenome, TdgClinicalTrial, TTD
PARP1 142 TALAZOPARIB TOSYLATE CHEMBL3137318 inhibitor ChemblInteractions
PARP1 142 OLAPARIB CHEMBL521686 inhibitor DrugBank, GuideToPharmacologyInteractions, MyCancerGenome, ClearityFoundationClinicalTrial, TTD, MyCancerGenomeClinicalTrial, ChemblInteractions 25981132

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID