Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
SCN11A 11280 PHENACEMIDE CHEMBL918 blocker ChemblInteractions
SCN11A 11280 CHLOROPROCAINE HYDROCHLORIDE CHEMBL944 blocker ChemblInteractions
SCN11A 11280 QUINIDINE GLUCONATE CHEMBL1200437 blocker ChemblInteractions
SCN11A 11280 PRIMIDONE CHEMBL856 blocker ChemblInteractions
SCN11A 11280 TOPIRAMATE CHEMBL220492 blocker ChemblInteractions
SCN11A 11280 RALFINAMIDE CHEMBL2107771 blocker ChemblInteractions
SCN11A 11280 TETRACAINE HYDROCHLORIDE CHEMBL1255654 blocker ChemblInteractions
SCN11A 11280 ESLICARBAZEPINE CHEMBL315985 blocker ChemblInteractions
SCN11A 11280 ETHOTOIN CHEMBL1095 blocker ChemblInteractions
SCN11A 11280 PROPOXYCAINE HYDROCHLORIDE CHEMBL1769 blocker ChemblInteractions
SCN11A 11280 LIDOCAINE CHEMBL79 blocker ChemblInteractions
SCN11A 11280 NW-3509 CHEMBL3545207 blocker ChemblInteractions
SCN11A 11280 HEXYLCAINE HYDROCHLORIDE CHEMBL1200715 blocker ChemblInteractions
SCN11A 11280 SAFINAMIDE CHEMBL396778 TdgClinicalTrial
SCN11A 11280 TETRODOTOXIN CHEMBL507974 TdgClinicalTrial
SCN11A 11280 QUINIDINE POLYGALACTURONATE CHEMBL1201486 blocker ChemblInteractions
SCN11A 11280 DISOPYRAMIDE PHOSPHATE CHEMBL1201020 blocker ChemblInteractions
SCN11A 11280 QUINIDINE SULFATE CHEMBL3707183 blocker ChemblInteractions
SCN11A 11280 ORPHENADRINE (CHLORIDE) CHEMBL1201023 blocker ChemblInteractions
SCN11A 11280 TOCAINIDE HYDROCHLORIDE CHEMBL1200773 blocker ChemblInteractions
SCN11A 11280 ESLICARBAZEPINE ACETATE CHEMBL87992 blocker ChemblInteractions
SCN11A 11280 ROPIVACAINE HYDROCHLORIDE CHEMBL1889140 blocker ChemblInteractions
SCN11A 11280 MEPHENYTOIN CHEMBL861 blocker ChemblInteractions
SCN11A 11280 PROCAINAMIDE HYDROCHLORIDE CHEMBL605 blocker ChemblInteractions
SCN11A 11280 PROPAFENONE HYDROCHLORIDE CHEMBL1201063 blocker ChemblInteractions
SCN11A 11280 PHENAZOPYRIDINE HYDROCHLORIDE CHEMBL1201022 blocker ChemblInteractions
SCN11A 11280 BENOXINATE HYDROCHLORIDE CHEMBL1200654 blocker ChemblInteractions
SCN11A 11280 MEXILETINE HYDROCHLORIDE CHEMBL1200606 blocker ChemblInteractions
SCN11A 11280 RILUZOLE CHEMBL744 blocker ChemblInteractions
SCN11A 11280 DRONEDARONE HYDROCHLORIDE CHEMBL1201729 blocker ChemblInteractions
SCN11A 11280 DYCLONINE HYDROCHLORIDE CHEMBL1200478 blocker ChemblInteractions
SCN11A 11280 PRILOCAINE CHEMBL1194 blocker ChemblInteractions
SCN11A 11280 PHENYTOIN SODIUM CHEMBL1611 blocker ChemblInteractions
SCN11A 11280 ETIDOCAINE HYDROCHLORIDE CHEMBL1200597 blocker ChemblInteractions
SCN11A 11280 OXCARBAZEPINE CHEMBL1068 blocker ChemblInteractions
SCN11A 11280 PHENYTOIN CHEMBL16 blocker ChemblInteractions
SCN11A 11280 FOSPHENYTOIN SODIUM CHEMBL919 blocker ChemblInteractions
SCN11A 11280 LAMOTRIGINE CHEMBL741 blocker ChemblInteractions
SCN11A 11280 NKTR-171 CHEMBL3545209 blocker ChemblInteractions
SCN11A 11280 MEPIVACAINE HYDROCHLORIDE CHEMBL1200440 blocker ChemblInteractions
SCN11A 11280 PRILOCAINE HYDROCHLORIDE CHEMBL1200586 blocker ChemblInteractions
SCN11A 11280 PROPARACAINE HYDROCHLORIDE CHEMBL1200464 blocker ChemblInteractions
SCN11A 11280 RUFINAMIDE CHEMBL1201754 blocker ChemblInteractions
SCN11A 11280 COCAINE CHEMBL370805 inhibitor TdgClinicalTrial, TEND, DrugBank 17139284, 17016423
SCN11A 11280 ZONISAMIDE CHEMBL750 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, DrugBank 19557119, 20025128, 20001433, 18433351, 14704463, 15511691, 19948168
SCN11A 11280 MERETHOXYLLINE PROCAINE CHEMBL1200443 blocker ChemblInteractions
SCN11A 11280 PROCAINE HYDROCHLORIDE CHEMBL1200841 blocker ChemblInteractions
SCN11A 11280 MORICIZINE HYDROCHLORIDE CHEMBL1200334 blocker ChemblInteractions
SCN11A 11280 INDECAINIDE HYDROCHLORIDE CHEMBL1200341 blocker ChemblInteractions
SCN11A 11280 LIDOCAINE HYDROCHLORIDE HYDRATE CHEMBL1200409 blocker ChemblInteractions
SCN11A 11280 Afacifenacin CHEMBL3545165 blocker ChemblInteractions
SCN11A 11280 NERISPIRDINE CHEMBL2107762 blocker ChemblInteractions
SCN11A 11280 ORPHENADRINE CITRATE CHEMBL1200395 blocker ChemblInteractions
SCN11A 11280 ARTICAINE HYDROCHLORIDE CHEMBL1200819 blocker ChemblInteractions
SCN11A 11280 TETRACAINE CHEMBL698 blocker ChemblInteractions
SCN11A 11280 CARBAMAZEPINE CHEMBL108 blocker ChemblInteractions
SCN11A 11280 LACOSAMIDE CHEMBL58323 blocker ChemblInteractions
SCN11A 11280 IRAMPANEL CHEMBL29741 blocker ChemblInteractions

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID