Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
TOP1 7150 CHEMBL343336 CHEMBL343336 DrugBank 10592235
TOP1 7150 ETIRINOTECAN PEGOL CHEMBL3039558 inhibitor ChemblInteractions
TOP1 7150 IRINOTECAN HYDROCHLORIDE HYDRATE CHEMBL1200512 inhibitor ChemblInteractions
TOP1 7150 ELSAMITRUCIN CHEMBL2106409 DrugBank
TOP1 7150 SODIUM STIBOGLUCONATE CHEMBL2079699 inhibitor DrugBank 15562618, 2835038, 10592235
TOP1 7150 BECATECARIN CHEMBL2107313 inhibitor ChemblInteractions
TOP1 7150 LURTOTECAN CHEMBL305666 TdgClinicalTrial
TOP1 7150 IRINOTECAN CHEMBL481 inhibitor ClearityFoundationBiomarkers, TdgClinicalTrial, ClearityFoundationClinicalTrial, CIViC, TEND, MyCancerGenomeClinicalTrial 19775480
TOP1 7150 TOPOTECAN CHEMBL84 ClearityFoundationBiomarkers, TdgClinicalTrial, ClearityFoundationClinicalTrial, TEND
TOP1 7150 C-1311 (CHEMBL3545337) CHEMBL3545337 TdgClinicalTrial
TOP1 7150 CAMPTOTHECIN CHEMBL65 TdgClinicalTrial, ClearityFoundationClinicalTrial, DrugBank 11752352, 18056711, 10592235, 18061144
TOP1 7150 EDOTECARIN CHEMBL435191 DrugBank 17325867, 15929804
TOP1 7150 LUCANTHONE CHEMBL279014 inhibitor DrugBank 10487533, 9169823
TOP1 7150 KARENITECIN CHEMBL1743260 TdgClinicalTrial, DrugBank
TOP1 7150 7-ETHYL-10-HYDROXY-CAMPTOTHECIN CHEMBL837 TdgClinicalTrial, DrugBank
TOP1 7150 CYCLOPHOSPHAMIDE CHEMBL88 NCI 1682037
TOP1 7150 IRINOTECAN SUCROSOFATE CHEMBL3039564 inhibitor ChemblInteractions
TOP1 7150 RUBITECAN CHEMBL77305 TdgClinicalTrial
TOP1 7150 CAFFEINE CHEMBL113 NCI 1339096

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID