Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
MTOR 2475 EVEROLIMUS CHEMBL1908360 inhibitor GuideToPharmacologyInteractions, CIViC, DrugBank, OncoKB, TTD, MyCancerGenome, TEND, TdgClinicalTrial, MyCancerGenomeClinicalTrial, ClearityFoundationClinicalTrial, TALC, CGI, DoCM 24625776, 25295501, 20569080, 20155724, 19774211, 11752352, 20531964, 19344392, 18466433, 27482884, 2015, 11010, 26859683, 24622468
MTOR 2475 CC-223 CHEMBL3545151 inhibitor GuideToPharmacologyInteractions, ChemblInteractions, CancerCommons
MTOR 2475 DACTOLISIB CHEMBL1879463 inhibitor GuideToPharmacologyInteractions, TALC, TTD, MyCancerGenome, MyCancerGenomeClinicalTrial, CancerCommons, ChemblInteractions
MTOR 2475 Palomid-529 CHEMBL2141712 inhibitor TdgClinicalTrial, ChemblInteractions
MTOR 2475 RG-7603 CHEMBL2331680 inhibitor ChemblInteractions
MTOR 2475 PWT-33579 CHEMBL3545323 inhibitor ChemblInteractions
MTOR 2475 CC-115 CHEMBL3545426 inhibitor ChemblInteractions
MTOR 2475 DS-7423 CHEMBL3545248 inhibitor ChemblInteractions
MTOR 2475 SIROLIMUS CHEMBL413 inhibitor OncoKB, ClearityFoundationClinicalTrial, DrugBank, TALC, MyCancerGenome, TTD, TdgClinicalTrial, CGI, CIViC, DoCM 27482884, 20005306, 11752352, 12742462, 19620795, 27279227, 24631838, 26619011
MTOR 2475 SF-1126 CHEMBL2326966 inhibitor MyCancerGenome, TdgClinicalTrial, ChemblInteractions, DrugBank
MTOR 2475 VOXTALISIB CHEMBL3545366 inhibitor TALC, MyCancerGenome, TdgClinicalTrial, ChemblInteractions, DrugBank, CancerCommons
MTOR 2475 TEMSIROLIMUS CHEMBL1201182 inhibitor MyCancerGenome, TEND, MyCancerGenomeClinicalTrial, DrugBank, GuideToPharmacologyInteractions, OncoKB, TALC, TdgClinicalTrial, TTD, CancerCommons, ClearityFoundationClinicalTrial 17935273, 11752352, 18265991, 27482884
MTOR 2475 GEDATOLISIB CHEMBL592445 inhibitor MyCancerGenome, GuideToPharmacologyInteractions, ChemblInteractions, MyCancerGenomeClinicalTrial
MTOR 2475 METFORMIN CHEMBL1431 inhibitor GuideToPharmacologyInteractions, MyCancerGenomeClinicalTrial
MTOR 2475 OMIPALISIB CHEMBL1236962 inhibitor GuideToPharmacologyInteractions, ChemblInteractions
MTOR 2475 RIDAFOROLIMUS CHEMBL2103839 inhibitor TALC, MyCancerGenome, TdgClinicalTrial, ClearityFoundationClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TTD
MTOR 2475 VS-5584 CHEMBL1079593 inhibitor GuideToPharmacologyInteractions, ChemblInteractions
MTOR 2475 CHEMBL561708 CHEMBL561708 inhibitor GuideToPharmacologyInteractions
MTOR 2475 DS-3078a CHEMBL3544963 inhibitor ChemblInteractions, CancerCommons
MTOR 2475 MLN-0128 CHEMBL3545097 inhibitor ChemblInteractions
MTOR 2475 PWT-33587 CHEMBL3545006 inhibitor ChemblInteractions
MTOR 2475 CHEMBL269259 CHEMBL269259 DrugBank
MTOR 2475 PA-799 CHEMBL1684984 inhibitor GuideToPharmacologyInteractions
MTOR 2475 LY-3023414 CHEMBL3544999 inhibitor GuideToPharmacologyInteractions, ChemblInteractions
MTOR 2475 SPARFLOXACIN CHEMBL850 inhibitor GuideToPharmacologyInteractions
MTOR 2475 TORIN1 CHEMBL1256459 inhibitor GuideToPharmacologyInteractions
MTOR 2475 BENZONATATE CHEMBL1374379 inhibitor GuideToPharmacologyInteractions
MTOR 2475 ALPELISIB CHEMBL2396661 inhibitor CancerCommons
MTOR 2475 PKI-179 CHEMBL1258517 inhibitor ChemblInteractions
MTOR 2475 BGT-226 (CHEMBL3545096) CHEMBL3545096 inhibitor ChemblInteractions
MTOR 2475 APITOLISIB CHEMBL1922094 inhibitor MyCancerGenome, GuideToPharmacologyInteractions, ChemblInteractions, TTD
MTOR 2475 INK-128 CHEMBL3545056 inhibitor MyCancerGenome, GuideToPharmacologyInteractions, ChemblInteractions, TTD
MTOR 2475 PF-04691502 CHEMBL1234354 inhibitor TALC, MyCancerGenome, GuideToPharmacologyInteractions, ChemblInteractions
MTOR 2475 PI-103 CHEMBL573339 inhibitor MyCancerGenome, GuideToPharmacologyInteractions
MTOR 2475 CHEMBL1081312 CHEMBL1081312 inhibitor GuideToPharmacologyInteractions
MTOR 2475 YOHIMBINE CHEMBL15245 inhibitor GuideToPharmacologyInteractions
MTOR 2475 OSI-027 CHEMBL3120215 inhibitor TALC, MyCancerGenome, TdgClinicalTrial, ChemblInteractions, TTD
MTOR 2475 Panulisib CHEMBL3545322 inhibitor ChemblInteractions
MTOR 2475 AZD-2014 CHEMBL1078983 inhibitor ChemblInteractions
MTOR 2475 AZD-8055 CHEMBL1801204 inhibitor TALC, MyCancerGenome, GuideToPharmacologyInteractions, ChemblInteractions, CIViC 27279227
MTOR 2475 PAZOPANIB CHEMBL477772 CIViC 24625776
MTOR 2475 AZD-5363 CHEMBL2178577 CIViC 26490311
MTOR 2475 PIMECROLIMUS CHEMBL1200686 potentiator TdgClinicalTrial, DrugBank 12113647
MTOR 2475 LY-294002 CHEMBL98350 CIViC 26490311

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID
MTOR rs12139042 GG carboplatin efficacy no No association was seen between this SNP and duration of progression free survival. Odds ratio below is for disease progression. Genotype GG is not associated with response to carboplatin or cisplatin in people with Carcinoma, Non-Small-Cell Lung as compared to genotypes AA + AG. 22901187 1183699216